ADAMTS-5 Inhibitor ( —— )

Catalog No. M26598 CAS No. 929634-33-3

ADAMTS-5 Inhibitor is a potent ADAMTS-5 (aggrecanase-2) inhibitor, with an IC50 of 1.1 μM. ADAMTS-5 Inhibitor shows >40-fold functional selectivity over ADAMTS-4 (aggrecanase-1).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	133	Get Quote
10MG	195	Get Quote
25MG	323	Get Quote
50MG	480	Get Quote
100MG	692	Get Quote
500MG	1422	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

ADAMTS-5 Inhibitor
Note

Research use only, not for human use.
Brief Description

ADAMTS-5 Inhibitor is a potent ADAMTS-5 (aggrecanase-2) inhibitor, with an IC50 of 1.1 μM. ADAMTS-5 Inhibitor shows >40-fold functional selectivity over ADAMTS-4 (aggrecanase-1).
Description

ADAMTS-5 Inhibitor is a potent ADAMTS-5 (aggrecanase-2) inhibitor, with an IC50 of 1.1 μM. ADAMTS-5 Inhibitor shows >40-fold functional selectivity over ADAMTS-4 (aggrecanase-1).
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

5-HT2A; D1 receptor; D5 receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

929634-33-3
Formula Weight

449.9
Molecular Formula

C16H11ClF3N3OS3
Purity

>98% (HPLC)
Solubility

——
SMILES

Cn1nc(c(\C=C2/SC(=S)NC2=O)c1SCc1ccc(Cl)cc1)C(F)(F)F
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.1. Rostom SA. Novel fused pyrrole heterocyclic ring systems as structure analogs of LE 300: Synthesis and pharmacological evaluation as serotonin 5-HT(2A), dopamine and histamine H(1) receptor ligands. Arch Pharm (Weinheim). 2010 Feb;343(2):73-80.

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